Presentations
OHE Tomoyuki
81-100 items (total 184)
Discovery and synthesis of a novel non-covalent inhibitor for protein-protein interaction between Nrf2 and Keap1
- Speaker
- Daisuke Yasuda, Tomoyuki Ohe, Rika Obata, Kyoko Takahashi, Tadahiko Mashino, Masaaki Komatsu, Yoshinobu Ichimura, Masayuki Yamamoto, Riyo Imamura, Hirotatsu Kojima, Takayoshi Okabe, Tetsuo Nagano
- Conference Title
- [Conference Category International presentation] Conference Title THE INTERNATIONAL CHEMICAL CONGRESS OF PACIFIC BASIN SOCIETIES 2015(Venue Honolulu, Hawaii, USA) Dates 2015.12.19 - 2015.12.19
- Presentation Format
- International presentation
- Language of Publication
- English
- Conference Category
- Poster presentation
Synthesis of multi-target fullerene derivatives with both HCV RNA polymerase inhibitory and antioxidant activities for the treatment of HCV-related disease
- Speaker
- Hiroki Kataoka, Kyoko Takahashi, Tomoyuki Ohe, Shigeo Nakamura, Tadahiko Mashino
- Conference Title
- [Conference Category International presentation] Conference Title THE INTERNATIONAL CHEMICAL CONGRESS OF PACIFIC BASIN SOCIETIES 2015(Venue Honolulu, Hawaii, USA) Dates 2015.12.16 - 2015.12.16
- Presentation Format
- International presentation
- Language of Publication
- English
- Conference Category
- Poster presentation
Synthesis of novel pyridine/pyridinium-type fullerene derivatives with human immunodeficiency virus-reverse transcriptase inhibition activity
- Speaker
- Takumi Yasuno, Kyoko Takahashi, Tomoyuki Ohe, Shigeo Nakamura, Tadahiko Mashino
- Conference Title
- [Conference Category International presentation] Conference Title THE INTERNATIONAL CHEMICAL CONGRESS OF PACIFIC BASIN SOCIETIES 2015(Venue Honolulu, Hawaii, USA) Dates 2015.12.16 - 2015.12.16
- Presentation Format
- International presentation
- Language of Publication
- English
- Conference Category
- Poster presentation
プロリン型フラーレン誘導体によるPPARγの活性阻害を介した脂肪細胞の分化抑制
- Speaker
- 服部 貴大, 多胡(船越) めぐみ, 大江 知之, 増野 匡彦, 田村 悦臣
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.12.01 - 2015.12.01
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
尿酸の構造を単純化した置換インドリノン誘導体の合成と抗酸化活性
- Speaker
- 高橋恭子,五十嵐拓,平石至,中村成夫,大江知之,増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.11.26 - 2015.11.26
- Organizer
- 日本薬学会 医薬化学部会
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
ベンズブロマロンの代謝物依存的なミトコンドリア毒性
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.11.12 - 2015.11.12
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
Novel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450
- Speaker
- Tomoyuki Ohe, Yumina Kitagawara, Kumiko Tachibana, Yuki Fujita, Kyoko Takahashi, Shigeo Nakamura, and Tadahiko Mashino
- Conference Title
- [Conference Category Domestic presentation] Conference Title 30th JSSX Annual Meeting(Venue Tokyo) Organizer JSSX Dates 2015.11.12 - 2015.11.12
- Organizer
- JSSX
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
インドール共役ヒダントイン誘導体の合成とラジカル消去活性
- Speaker
- 岡崎希望、槇田智史、高橋恭子、大江知之、中村成夫、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.09.12 - 2015.09.12
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
抗酸化活性環状ジペプチド化合物の脂質過酸化抑制効果
- Speaker
- 槇田 智史, 高橋 恭子, 池 貴幸, 安田 大輔, 中村 成夫, 大江 知之, 増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.06.12 - 2015.06.12
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
C-4 位メチル基が関与するnevirapineの代謝活性化機構の解析
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.03.28 - 2015.03.28
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
新規抗酸化剤環状 arylvinyl alcohol 類のデザインと合成
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.03.28 - 2015.03.28
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
HCV RNAポリメラーゼ阻害活性を有する新規プロリン型フラーレン誘導体の創製
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.03.28 - 2015.03.28
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
Cyclooxygenase (COX) 阻害作用を持たないmeloxicam類縁体も MPP+誘発SH-SY5Y神経細胞死を抑制する
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.03.27 - 2015.03.27
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
チオラクタム構造を経由した新規水溶性フラーレン誘導体の合成とその脂質過酸化抑制効果
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.03.27 - 2015.03.27
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
多標的型 AIDS 関連疾患治療薬を目指した 5-(methylpyridinium)proline 型フラーレン誘導体の構造変換
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.03.27 - 2015.03.27
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
慶應義塾創立 150 年記念未来先導基金 慶應義塾大学薬学部「国際医薬品開発と規制を先導する薬学人材育成プログラム」
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2015.03.26 - 2015.03.26
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
Synthesis and biological evaluation of novel nevirapine analogs designed to avoid metabolic activation
- Speaker
- Yasuhiro Tateishi, Tomoyuki Ohe, Kyoko Takahashi, Shigeo Nakamura, Tadahiko Mashino
- Conference Title
- [Conference Category International presentation] Dates 2018.10.04 - 2018.10.04
- Presentation Format
- International presentation
- Language of Publication
- English
- Conference Category
- Poster presentation
新規アザフレロイド誘導体の合成と HCV RNA ポリメラーゼ阻害活性
- Speaker
- 薮内大貴、片岡裕樹、高橋 恭子、中村 成夫、大江 知之、増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2018.09.15 - 2018.09.15
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
がん細胞増殖抑制効果を有するカチオン型フラーレン誘導体による活性酸素産生およびその構造活性相関
- Speaker
- 池田 瞳、安田 大輔、高橋 恭子、中村 成夫、大江 知之、増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2018.09.15 - 2018.09.15
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
Synthesis of a fluoroalkene mimic of an amide drug via copper-catalyzed defluoroborylation and evaluation of its properties
- Speaker
- Takashi Niwa, Yuta Uetake, Motoyuki Isoda, Tomoyuki Ohe, Daisuke Yasuda, Tadahiko Mashino, Takamitsu Hosoya
- Conference Title
- [Conference Category Domestic presentation] Conference Title The 13th Annual Meeting of Japanese Society for Chemical Biology Dates 2018.06.12 - 2018.06.12
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation