Keio University

Presentations

OHE Tomoyuki

81-100 items (total 184)

Discovery and synthesis of a novel non-covalent inhibitor for protein-protein interaction between Nrf2 and Keap1

Speaker
Daisuke Yasuda, Tomoyuki Ohe, Rika Obata, Kyoko Takahashi, Tadahiko Mashino, Masaaki Komatsu, Yoshinobu Ichimura, Masayuki Yamamoto, Riyo Imamura, Hirotatsu Kojima, Takayoshi Okabe, Tetsuo Nagano
Conference Title
[Conference Category International presentation] Conference Title THE INTERNATIONAL CHEMICAL CONGRESS OF PACIFIC BASIN SOCIETIES 2015(Venue Honolulu, Hawaii, USA) Dates 2015.12.19 - 2015.12.19
Presentation Format
International presentation
Language of Publication
English
Conference Category
Poster presentation

Synthesis of multi-target fullerene derivatives with both HCV RNA polymerase inhibitory and antioxidant activities for the treatment of HCV-related disease

Speaker
Hiroki Kataoka, Kyoko Takahashi, Tomoyuki Ohe, Shigeo Nakamura, Tadahiko Mashino
Conference Title
[Conference Category International presentation] Conference Title THE INTERNATIONAL CHEMICAL CONGRESS OF PACIFIC BASIN SOCIETIES 2015(Venue Honolulu, Hawaii, USA) Dates 2015.12.16 - 2015.12.16
Presentation Format
International presentation
Language of Publication
English
Conference Category
Poster presentation

Synthesis of novel pyridine/pyridinium-type fullerene derivatives with human immunodeficiency virus-reverse transcriptase inhibition activity

Speaker
Takumi Yasuno, Kyoko Takahashi, Tomoyuki Ohe, Shigeo Nakamura, Tadahiko Mashino
Conference Title
[Conference Category International presentation] Conference Title THE INTERNATIONAL CHEMICAL CONGRESS OF PACIFIC BASIN SOCIETIES 2015(Venue Honolulu, Hawaii, USA) Dates 2015.12.16 - 2015.12.16
Presentation Format
International presentation
Language of Publication
English
Conference Category
Poster presentation

プロリン型フラーレン誘導体によるPPARγの活性阻害を介した脂肪細胞の分化抑制

Speaker
服部 貴大, 多胡(船越) めぐみ, 大江 知之, 増野 匡彦, 田村 悦臣
Conference Title
[Conference Category Domestic presentation] Dates 2015.12.01 - 2015.12.01
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

尿酸の構造を単純化した置換インドリノン誘導体の合成と抗酸化活性

Speaker
高橋恭子,五十嵐拓,平石至,中村成夫,大江知之,増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2015.11.26 - 2015.11.26
Organizer
日本薬学会 医薬化学部会
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

ベンズブロマロンの代謝物依存的なミトコンドリア毒性

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.11.12 - 2015.11.12
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

Novel Bioactivation Pathway of Benzbromarone Mediated by Cytochrome P450

Speaker
Tomoyuki Ohe, Yumina Kitagawara, Kumiko Tachibana, Yuki Fujita, Kyoko Takahashi, Shigeo Nakamura, and Tadahiko Mashino
Conference Title
[Conference Category Domestic presentation] Conference Title 30th JSSX Annual Meeting(Venue Tokyo) Organizer JSSX Dates 2015.11.12 - 2015.11.12
Organizer
JSSX
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

インドール共役ヒダントイン誘導体の合成とラジカル消去活性

Speaker
岡崎希望、槇田智史、高橋恭子、大江知之、中村成夫、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2015.09.12 - 2015.09.12
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

抗酸化活性環状ジペプチド化合物の脂質過酸化抑制効果

Speaker
槇田 智史, 高橋 恭子, 池 貴幸, 安田 大輔, 中村 成夫, 大江 知之, 増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2015.06.12 - 2015.06.12
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

C-4 位メチル基が関与するnevirapineの代謝活性化機構の解析

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.03.28 - 2015.03.28
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

新規抗酸化剤環状 arylvinyl alcohol 類のデザインと合成

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.03.28 - 2015.03.28
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

HCV RNAポリメラーゼ阻害活性を有する新規プロリン型フラーレン誘導体の創製

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.03.28 - 2015.03.28
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

Cyclooxygenase (COX) 阻害作用を持たないmeloxicam類縁体も MPP+誘発SH-SY5Y神経細胞死を抑制する

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.03.27 - 2015.03.27
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

チオラクタム構造を経由した新規水溶性フラーレン誘導体の合成とその脂質過酸化抑制効果

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.03.27 - 2015.03.27
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

多標的型 AIDS 関連疾患治療薬を目指した 5-(methylpyridinium)proline 型フラーレン誘導体の構造変換

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.03.27 - 2015.03.27
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

慶應義塾創立 150 年記念未来先導基金 慶應義塾大学薬学部「国際医薬品開発と規制を先導する薬学人材育成プログラム」

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2015.03.26 - 2015.03.26
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

Synthesis and biological evaluation of novel nevirapine analogs designed to avoid metabolic activation

Speaker
Yasuhiro Tateishi, Tomoyuki Ohe, Kyoko Takahashi, Shigeo Nakamura, Tadahiko Mashino
Conference Title
[Conference Category International presentation] Dates 2018.10.04 - 2018.10.04
Presentation Format
International presentation
Language of Publication
English
Conference Category
Poster presentation

新規アザフレロイド誘導体の合成と HCV RNA ポリメラーゼ阻害活性

Speaker
薮内大貴、片岡裕樹、高橋 恭子、中村 成夫、大江 知之、増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.09.15 - 2018.09.15
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

がん細胞増殖抑制効果を有するカチオン型フラーレン誘導体による活性酸素産生およびその構造活性相関

Speaker
池田 瞳、安田 大輔、高橋 恭子、中村 成夫、大江 知之、増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.09.15 - 2018.09.15
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

Synthesis of a fluoroalkene mimic of an amide drug via copper-catalyzed defluoroborylation and evaluation of its properties

Speaker
Takashi Niwa, Yuta Uetake, Motoyuki Isoda, Tomoyuki Ohe, Daisuke Yasuda, Tadahiko Mashino, Takamitsu Hosoya
Conference Title
[Conference Category Domestic presentation] Conference Title The 13th Annual Meeting of Japanese Society for Chemical Biology Dates 2018.06.12 - 2018.06.12
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation