Keio University

Presentations

OHE Tomoyuki

41-60 items (total 184)

Synthesis and evaluation of novel diclofenac analogues to mitigate its metabolic activation via glucuronidation

Speaker
Yasuhiro Tateishi , Tomoyuki Ohe , Daisuke Yasuda , Kyoko Takahashi , Shigeo Nakamura , Tadahiko Mashino
Conference Title
[Conference Category Domestic presentation] Dates 2019.12.10 - 2019.12.10
Presentation Format
Domestic presentation
Language of Publication
English
Conference Category
Oral presentation (general)

Development of a novel method to detect reactive metabolites – Synthesis of fluorescent-labeled trapping reagents based on cysteine and assessment of their reactivities –

Speaker
Chikako Shibazaki, Kyoko Takahashi, Shigeo Nakamura, Tomoyuki Ohe, Tadahiko Mashino
Conference Title
[Conference Category Domestic presentation] Dates 2019.11.27 - 2019.11.27
Presentation Format
Domestic presentation
Language of Publication
English
Conference Category
Poster presentation

HIV プロテアーゼ阻害活性を有するプロリン型フラーレン誘導体の立体選択的合成

Speaker
片岸大紀, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.09.14 - 2019.09.14
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

リモナバンの代謝活性化を回避する構造変換

Speaker
除川貴太, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.09.14 - 2019.09.14
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

Wntシグナル抑制によりウイルス感染非ホジキンリンパ腫の細胞増殖を抑制するフラーレン誘導体の開発

Speaker
門田彩乃,森口美里,渡部匡史,中村成夫,安野拓実,大江知之,増野匡彦,藤室雅弘
Conference Title
[Conference Category Domestic presentation] Dates 2020.03.27 - 2020.03.27
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

トラッピング剤を用いた反応性アシルグルクロニドの新規検出法

Speaker
柴﨑 智香子, 高橋 恭子, 中村成夫, 大江 知之, 増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2020.03.26 - 2020.03.26
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

HIV/HCV共感染治療薬を志向した 多標的型ピリジニウム型C60誘導体の創製

Speaker
小林透威, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2020.03.27 - 2020.03.27
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

代謝活性化回避を指向した新規ジクロフェナク類縁体の合成と評価

Speaker
立石泰寛, 大江知之, 小川真依, 安田大輔, 高橋恭子, 中村成夫, 増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2020.03.28 - 2020.03.28
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

抗がん活性を有するカチオン型C60誘導体のミトコンドリア機能障害

Speaker
高橋恭子,池田瞳,安田大輔,中村成夫,大江知之,増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.06.27 - 2019.06.27
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

ハード及びソフトな反応性代謝物を捕捉する新規蛍光標識トラッピング剤の創製

Speaker
柴崎智香子、髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

オキシカム構造を模倣したスルホン類の抗パーキンソン病効果

Speaker
小町元輝、鈴木啓太、高橋恭子、中村成夫、大江知之、大久保知子、春名柚佳、田﨑嘉一、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

ハードな反応性代謝物を捕捉する新規蛍光標識化トラッピング剤の創製

Speaker
長邑花、柴崎智香子、髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

フッ素導入により反応性代謝物の生成を回避した改良型Diclofenac類縁体の創製

Speaker
小川 真依、山田晶子、安田大輔、高橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

p62-Keap1-Nrf2系を標的としたPPI阻害剤の幹細胞がん薬剤耐性抑制効果

Speaker
安田大輔、大江知之、高橋恭子、小松雅明、一村義信、山本雅之、今村理世、小島宏建、岡部隆義、長野哲雄、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.11.29 - 2018.11.29
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

抗パーキンソン病活性を有するテトラロンアナログB環へのフッ素の導入と神経細胞保護効果

Speaker
伊藤廉、梅本英明、三山由茉子、高橋恭子、中村成夫、大江知之、大久保知子、春名柚佳、田﨑嘉一、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

ピリジニウム型フラーレン誘導体のウイルス感染リンパ腫に対する抗腫瘍活性

Speaker
門田 彩乃, 森口 美里、 渡部 匡史、中村 成夫、安野 拓実、 大江 知之、 増野 匡彦 、藤室 雅弘
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

HIVプロテアーゼおよび逆転写酵素阻害活性を有する新規多標的型C60誘導体の創製:基質遷移状態模倣型イソスターとC60コアを結ぶリンカーの長さの検討

Speaker
古川 慶吾、髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

ADMET研究と創薬化学を融合した新しいアカデミア創薬

Speaker
OHE Tomoyuki
Conference Title
[Conference Category Domestic presentation] Dates 2017.09.16 - 2017.09.16
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Symposium, workshop panel (nominated)

抗がん薬を⽬指した新規ピリジニウム型C60 誘導体の創製

Speaker
安野拓実, ⾼橋恭⼦,大江知之, 中村成夫, 渡部匡史, 藤室雅弘, 増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2017.09.12 - 2017.09.12
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

HIV逆転写酵素及びプロテアーゼを阻害する多標的型新規フラーレン誘導体の創製

Speaker
橋本 航匠, 片岡 裕樹, 加藤 舞, 秋葉 智紘, 安野 拓実, 高橋 恭子, 大江 知 之, 中村 成夫, 増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2017.03.27 - 2017.03.27
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation