Presentations
OHE Tomoyuki
41-60 items (total 184)
Synthesis and evaluation of novel diclofenac analogues to mitigate its metabolic activation via glucuronidation
- Speaker
- Yasuhiro Tateishi , Tomoyuki Ohe , Daisuke Yasuda , Kyoko Takahashi , Shigeo Nakamura , Tadahiko Mashino
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.12.10 - 2019.12.10
- Presentation Format
- Domestic presentation
- Language of Publication
- English
- Conference Category
- Oral presentation (general)
Development of a novel method to detect reactive metabolites – Synthesis of fluorescent-labeled trapping reagents based on cysteine and assessment of their reactivities –
- Speaker
- Chikako Shibazaki, Kyoko Takahashi, Shigeo Nakamura, Tomoyuki Ohe, Tadahiko Mashino
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.11.27 - 2019.11.27
- Presentation Format
- Domestic presentation
- Language of Publication
- English
- Conference Category
- Poster presentation
HIV プロテアーゼ阻害活性を有するプロリン型フラーレン誘導体の立体選択的合成
- Speaker
- 片岸大紀, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.09.14 - 2019.09.14
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
リモナバンの代謝活性化を回避する構造変換
- Speaker
- 除川貴太, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.09.14 - 2019.09.14
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
Wntシグナル抑制によりウイルス感染非ホジキンリンパ腫の細胞増殖を抑制するフラーレン誘導体の開発
- Speaker
- 門田彩乃,森口美里,渡部匡史,中村成夫,安野拓実,大江知之,増野匡彦,藤室雅弘
- Conference Title
- [Conference Category Domestic presentation] Dates 2020.03.27 - 2020.03.27
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
トラッピング剤を用いた反応性アシルグルクロニドの新規検出法
- Speaker
- 柴﨑 智香子, 高橋 恭子, 中村成夫, 大江 知之, 増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2020.03.26 - 2020.03.26
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
HIV/HCV共感染治療薬を志向した 多標的型ピリジニウム型C60誘導体の創製
- Speaker
- 小林透威, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2020.03.27 - 2020.03.27
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
代謝活性化回避を指向した新規ジクロフェナク類縁体の合成と評価
- Speaker
- 立石泰寛, 大江知之, 小川真依, 安田大輔, 高橋恭子, 中村成夫, 増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2020.03.28 - 2020.03.28
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
抗がん活性を有するカチオン型C60誘導体のミトコンドリア機能障害
- Speaker
- 高橋恭子,池田瞳,安田大輔,中村成夫,大江知之,増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.06.27 - 2019.06.27
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
ハード及びソフトな反応性代謝物を捕捉する新規蛍光標識トラッピング剤の創製
- Speaker
- 柴崎智香子、髙橋恭子、中村成夫、大江知之、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
オキシカム構造を模倣したスルホン類の抗パーキンソン病効果
- Speaker
- 小町元輝、鈴木啓太、高橋恭子、中村成夫、大江知之、大久保知子、春名柚佳、田﨑嘉一、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
ハードな反応性代謝物を捕捉する新規蛍光標識化トラッピング剤の創製
- Speaker
- 長邑花、柴崎智香子、髙橋恭子、中村成夫、大江知之、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
フッ素導入により反応性代謝物の生成を回避した改良型Diclofenac類縁体の創製
- Speaker
- 小川 真依、山田晶子、安田大輔、高橋恭子、中村成夫、大江知之、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
p62-Keap1-Nrf2系を標的としたPPI阻害剤の幹細胞がん薬剤耐性抑制効果
- Speaker
- 安田大輔、大江知之、高橋恭子、小松雅明、一村義信、山本雅之、今村理世、小島宏建、岡部隆義、長野哲雄、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2018.11.29 - 2018.11.29
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
抗パーキンソン病活性を有するテトラロンアナログB環へのフッ素の導入と神経細胞保護効果
- Speaker
- 伊藤廉、梅本英明、三山由茉子、高橋恭子、中村成夫、大江知之、大久保知子、春名柚佳、田﨑嘉一、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
ピリジニウム型フラーレン誘導体のウイルス感染リンパ腫に対する抗腫瘍活性
- Speaker
- 門田 彩乃, 森口 美里、 渡部 匡史、中村 成夫、安野 拓実、 大江 知之、 増野 匡彦 、藤室 雅弘
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
HIVプロテアーゼおよび逆転写酵素阻害活性を有する新規多標的型C60誘導体の創製:基質遷移状態模倣型イソスターとC60コアを結ぶリンカーの長さの検討
- Speaker
- 古川 慶吾、髙橋恭子、中村成夫、大江知之、増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2019.03.21 - 2019.03.21
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
ADMET研究と創薬化学を融合した新しいアカデミア創薬
- Speaker
- OHE Tomoyuki
- Conference Title
- [Conference Category Domestic presentation] Dates 2017.09.16 - 2017.09.16
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Symposium, workshop panel (nominated)
抗がん薬を⽬指した新規ピリジニウム型C60 誘導体の創製
- Speaker
- 安野拓実, ⾼橋恭⼦,大江知之, 中村成夫, 渡部匡史, 藤室雅弘, 増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2017.09.12 - 2017.09.12
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
HIV逆転写酵素及びプロテアーゼを阻害する多標的型新規フラーレン誘導体の創製
- Speaker
- 橋本 航匠, 片岡 裕樹, 加藤 舞, 秋葉 智紘, 安野 拓実, 高橋 恭子, 大江 知 之, 中村 成夫, 増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2017.03.27 - 2017.03.27
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation