Keio University

Presentations

OHE Tomoyuki

21-40 items (total 184)

ADMET研究への有機化学的アプローチ

Speaker
大江知之
Conference Title
[Conference Category Domestic presentation] Dates 2021.07.19 - 2021.07.19
Invitation Status
With
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Public lecture, seminar, tutorial, course, or other speech
2022.03

パーキンソン病治療薬を目指したオキシカムアナログのADME評価および類縁体合成

Speaker
鶴岡 航太朗、高橋 恭子、中村 成夫、熊谷 直哉、増野 匡彦、大久保 知子、眞鍋 貴行、田﨑 嘉一、大江 知之
Conference Title
[Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
International Co-authorship
No
Conference Category
Oral presentation (general)
2022.11

オキシカム系抗炎症薬を基盤にした抗パーキンソン病薬の創製研究

Speaker
大江知之
Conference Title
[Conference Category Domestic presentation] Dates 2022.11.07 - 2022.11.10
Invitation Status
With
Presentation Format
Domestic presentation
Language of Publication
English
International Co-authorship
No
Conference Category
Symposium, workshop panel (nominated)
2022.03

ビスピリジニウム型フラーレン誘導体によるBCR-ABL陽性K562細胞のアポトーシス誘導機構の解析

Speaker
鷲見 和也、多胡 憲治、中澤 洋介、高橋 恭子、大江 知之、増野 匡彦、多胡 めぐみ
Conference Title
[Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
International Co-authorship
No
Conference Category
Oral presentation (general)
2022.03

マロン酸型フラーレン誘導体はSARS-CoV-2メインプロテアーゼを強く阻害する

Speaker
片岸 大紀、岩﨑 彩希子、安田 大輔、高橋 恭子、中村 成夫、増野 匡彦、熊谷 直哉、大江 知之
Conference Title
[Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
International Co-authorship
No
Conference Category
Oral presentation (general)
2022.03

胆道がん治療薬を目指したフェンチコナゾール誘導体の合成と評価

Speaker
木原 和輝、柏木 伸章、村松 俊英、高橋 恭子、中村 成夫、熊谷 直哉、増野 匡彦、齋藤 義正、大江 知之
Conference Title
[Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
International Co-authorship
No
Conference Category
Oral presentation (general)
2022.03

ヒト肝細胞を用いたトラッピング試験系の確立とその評価

Speaker
柴崎 智香子、増野 匡彦、熊谷 直哉、大江 知之
Conference Title
[Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
International Co-authorship
No
Conference Category
Oral presentation (general)

Development of fluorescent-labeled trapping reagents based on cysteine for detecting reactive metabolites

Speaker
Shibazaki C., Takahashi K., Nakamura S., Mashino T., Ohe T.
Conference Title
[Conference Category International presentation] Conference Title Pacifichem 2021 Dates 2021.12.19 - 2021.12.19
Invitation Status
Without
Presentation Format
International presentation
Language of Publication
Japanese
Conference Category
Poster presentation

Stereoselective synthesis and evaluation of fullerene derivatives as antiviral drugs

Speaker
Katagishi D., Takahashi K., Nakamura S., Mashino T., Ohe T.
Conference Title
[Conference Category International presentation] Conference Title Pacifichem 2021(Venue Hawaii (Online)) Dates 2021.12.20 - 2021.12.20
Presentation Format
International presentation
Language of Publication
English
Conference Category
Poster presentation

創薬における反応性代謝物のリスク評価

Speaker
大江知之
Conference Title
[Conference Category Domestic presentation] Dates 2017.01 - 2017.01
Invitation Status
With
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Public lecture, seminar, tutorial, course, or other speech

医薬品開発における反応性代謝物の評価

Speaker
大江知之
Conference Title
[Conference Category Domestic presentation] Dates 2012.03 - 2012.03
Invitation Status
With
Presentation Format
Domestic presentation
Language of Publication
English
Conference Category
Public lecture, seminar, tutorial, course, or other speech

TC-HepG2 細胞を用いた反応性代謝物の毒性評価と創薬への応用

Speaker
大江知之
Conference Title
[Conference Category Domestic presentation] Dates 2021.09.24 - 2021.09.24
Invitation Status
With
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Public lecture, seminar, tutorial, course, or other speech

Nrf2活性を制御するタンパク質間相互作用阻害剤の創成

Speaker
安田大輔, 今村理世, 小島宏建, 岡部隆義, 高橋恭子, 熊谷直哉,一村義信, 小松雅明, 山本雅之, 長野哲雄, 増野匡彦, 大江知之
Conference Title
[Conference Category Domestic presentation] Dates 2021.06.21 - 2021.06.21
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

p62-Keap1-Nrf2 系を標的とした抗がん剤感受性増強剤の創製

Speaker
安田大輔, 吉田逸平, 高橋恭子, 熊谷直哉, 増野匡彦, 今村理世, 小島宏建, 岡部隆義, 一村義信, 小松雅明, 山本雅之, 長野哲雄, 大江知之
Conference Title
[Conference Category Domestic presentation] Dates 2021.05.19 - 2021.05.19
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

抗パーキンソン病薬を目指した新規オキシカムA環芳香族複素環アナログの創製

Speaker
鶴岡 航太朗、小町 元輝、鈴木 啓太、高橋 恭子、中村 成夫、大江 知之、大久保 知子、眞鍋 貴之、田﨑 嘉一、増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2021.03.28 - 2021.03.28
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

シトクロムP450による5-置換-2-オキシインドールのipso置換代謝反応

Speaker
公平 実希、大江 知之、高橋 恭子、中村 成夫、増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2021.03.27 - 2021.03.27
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

反応性の高いアシルグルクロニドを検出する新規蛍光標識トラッピング剤の創製

Speaker
柴﨑 智香子、大江 知之、高橋 恭子、中村 成夫、増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2021.03.27 - 2021.03.27
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

代謝活性化の回避を目指したトファシチニブ類縁体の合成と評価

Speaker
立石 泰寛、大江 知之、高橋 恭子、中村 成夫、増野 匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2021.03.28 - 2021.03.28
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

HIVプロテアーゼ/逆転写酵素、HCV NS5B を標的とするピリジニウム型C60誘導体の創製

Speaker
小林透威, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2020.09.19 - 2020.09.19
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

新規抗血小板薬NSP-513のヒト, ラットおよびイヌにおけるin vitro代謝 酸化開裂型代謝物の同定とヒトの代謝におけるCYP3A4の関与

Speaker
石原 亜矢, 石井 康行, 柴田 芳宏, 大江 知之, 安盛 俊雄, 亀井 敏夫
Conference Title
[Conference Category Domestic presentation] Dates 1998.11.20 - 1998.11.20
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)