Presentations
OHE Tomoyuki
21-40 items (total 184)
ADMET研究への有機化学的アプローチ
- Speaker
- 大江知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.07.19 - 2021.07.19
- Invitation Status
- With
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Public lecture, seminar, tutorial, course, or other speech
2022.03
パーキンソン病治療薬を目指したオキシカムアナログのADME評価および類縁体合成
- Speaker
- 鶴岡 航太朗、高橋 恭子、中村 成夫、熊谷 直哉、増野 匡彦、大久保 知子、眞鍋 貴行、田﨑 嘉一、大江 知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- International Co-authorship
- No
- Conference Category
- Oral presentation (general)
2022.11
オキシカム系抗炎症薬を基盤にした抗パーキンソン病薬の創製研究
- Speaker
- 大江知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2022.11.07 - 2022.11.10
- Invitation Status
- With
- Presentation Format
- Domestic presentation
- Language of Publication
- English
- International Co-authorship
- No
- Conference Category
- Symposium, workshop panel (nominated)
2022.03
ビスピリジニウム型フラーレン誘導体によるBCR-ABL陽性K562細胞のアポトーシス誘導機構の解析
- Speaker
- 鷲見 和也、多胡 憲治、中澤 洋介、高橋 恭子、大江 知之、増野 匡彦、多胡 めぐみ
- Conference Title
- [Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- International Co-authorship
- No
- Conference Category
- Oral presentation (general)
2022.03
マロン酸型フラーレン誘導体はSARS-CoV-2メインプロテアーゼを強く阻害する
- Speaker
- 片岸 大紀、岩﨑 彩希子、安田 大輔、高橋 恭子、中村 成夫、増野 匡彦、熊谷 直哉、大江 知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- International Co-authorship
- No
- Conference Category
- Oral presentation (general)
2022.03
胆道がん治療薬を目指したフェンチコナゾール誘導体の合成と評価
- Speaker
- 木原 和輝、柏木 伸章、村松 俊英、高橋 恭子、中村 成夫、熊谷 直哉、増野 匡彦、齋藤 義正、大江 知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- International Co-authorship
- No
- Conference Category
- Oral presentation (general)
2022.03
ヒト肝細胞を用いたトラッピング試験系の確立とその評価
- Speaker
- 柴崎 智香子、増野 匡彦、熊谷 直哉、大江 知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2022.03.25 - 2022.03.28
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- International Co-authorship
- No
- Conference Category
- Oral presentation (general)
Development of fluorescent-labeled trapping reagents based on cysteine for detecting reactive metabolites
- Speaker
- Shibazaki C., Takahashi K., Nakamura S., Mashino T., Ohe T.
- Conference Title
- [Conference Category International presentation] Conference Title Pacifichem 2021 Dates 2021.12.19 - 2021.12.19
- Invitation Status
- Without
- Presentation Format
- International presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
Stereoselective synthesis and evaluation of fullerene derivatives as antiviral drugs
- Speaker
- Katagishi D., Takahashi K., Nakamura S., Mashino T., Ohe T.
- Conference Title
- [Conference Category International presentation] Conference Title Pacifichem 2021(Venue Hawaii (Online)) Dates 2021.12.20 - 2021.12.20
- Presentation Format
- International presentation
- Language of Publication
- English
- Conference Category
- Poster presentation
創薬における反応性代謝物のリスク評価
- Speaker
- 大江知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2017.01 - 2017.01
- Invitation Status
- With
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Public lecture, seminar, tutorial, course, or other speech
医薬品開発における反応性代謝物の評価
- Speaker
- 大江知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2012.03 - 2012.03
- Invitation Status
- With
- Presentation Format
- Domestic presentation
- Language of Publication
- English
- Conference Category
- Public lecture, seminar, tutorial, course, or other speech
TC-HepG2 細胞を用いた反応性代謝物の毒性評価と創薬への応用
- Speaker
- 大江知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.09.24 - 2021.09.24
- Invitation Status
- With
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Public lecture, seminar, tutorial, course, or other speech
Nrf2活性を制御するタンパク質間相互作用阻害剤の創成
- Speaker
- 安田大輔, 今村理世, 小島宏建, 岡部隆義, 高橋恭子, 熊谷直哉,一村義信, 小松雅明, 山本雅之, 長野哲雄, 増野匡彦, 大江知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.06.21 - 2021.06.21
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Poster presentation
p62-Keap1-Nrf2 系を標的とした抗がん剤感受性増強剤の創製
- Speaker
- 安田大輔, 吉田逸平, 高橋恭子, 熊谷直哉, 増野匡彦, 今村理世, 小島宏建, 岡部隆義, 一村義信, 小松雅明, 山本雅之, 長野哲雄, 大江知之
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.05.19 - 2021.05.19
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
抗パーキンソン病薬を目指した新規オキシカムA環芳香族複素環アナログの創製
- Speaker
- 鶴岡 航太朗、小町 元輝、鈴木 啓太、高橋 恭子、中村 成夫、大江 知之、大久保 知子、眞鍋 貴之、田﨑 嘉一、増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.03.28 - 2021.03.28
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
シトクロムP450による5-置換-2-オキシインドールのipso置換代謝反応
- Speaker
- 公平 実希、大江 知之、高橋 恭子、中村 成夫、増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.03.27 - 2021.03.27
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
反応性の高いアシルグルクロニドを検出する新規蛍光標識トラッピング剤の創製
- Speaker
- 柴﨑 智香子、大江 知之、高橋 恭子、中村 成夫、増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.03.27 - 2021.03.27
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
代謝活性化の回避を目指したトファシチニブ類縁体の合成と評価
- Speaker
- 立石 泰寛、大江 知之、高橋 恭子、中村 成夫、増野 匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2021.03.28 - 2021.03.28
- Invitation Status
- Without
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
HIVプロテアーゼ/逆転写酵素、HCV NS5B を標的とするピリジニウム型C60誘導体の創製
- Speaker
- 小林透威, 高橋恭子, 中村成夫, 大江知之, 増野匡彦
- Conference Title
- [Conference Category Domestic presentation] Dates 2020.09.19 - 2020.09.19
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)
新規抗血小板薬NSP-513のヒト, ラットおよびイヌにおけるin vitro代謝 酸化開裂型代謝物の同定とヒトの代謝におけるCYP3A4の関与
- Speaker
- 石原 亜矢, 石井 康行, 柴田 芳宏, 大江 知之, 安盛 俊雄, 亀井 敏夫
- Conference Title
- [Conference Category Domestic presentation] Dates 1998.11.20 - 1998.11.20
- Presentation Format
- Domestic presentation
- Language of Publication
- Japanese
- Conference Category
- Oral presentation (general)