Keio University

Presentations

Mashino, Tadahiko

41-60 items (total 386)

ハードな反応性代謝物を捕捉する新規蛍光標識化トラッピング剤の創製

Speaker
長邑花、柴崎智香子、髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
Dates 2019.03.20 - 2019.03.20
Language of Publication
Japanese

オキシカム構造を模倣したスルホン類の抗パーキンソン病効果

Speaker
小町元輝、鈴木啓太、高橋恭子、中村成夫、大江知之、大久保知子、春名柚佳、田﨑嘉一、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.20 - 2019.03.20
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

ハード及びソフトな反応性代謝物を捕捉する新規蛍光標識トラッピング剤の創製

Speaker
柴崎智香子、髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2019.03.20 - 2019.03.20
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

p62-Keap1-Nrf2系を標的としたPPI阻害剤の幹細胞がん薬剤耐性抑制効果

Speaker
安田大輔、大江知之、高橋恭子、小松雅明、一村義信、山本雅之、今村理世、小島宏建、岡部隆義、長野哲雄、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.11.28 - 2018.11.28
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

Synthesis and biological evaluation of novel nevirapine analogs designed to avoid metabolic activation

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category International presentation] Conference Title 2018 International Meeting on 22nd MDO and 33rd JSSX Dates 2018.10.04 - 2018.10.04
Presentation Format
International presentation
Language of Publication
English
Conference Category
Poster presentation

新規アザフレロイド誘導体の合成と HCV RNA ポリメラーゼ阻害活性

Speaker
○藪内大貴、片岡裕樹、髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.09.15 - 2018.09.15
Organizer
第62回日本薬学会関東支部大会
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

がん細胞増殖抑制効果を有するカチオン型フラーレン誘導体による活性酸素産生およびその構造活性相関

Speaker
○池田瞳、安田大輔、髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.09.15 - 2018.09.15
Organizer
第62回日本薬学会関東支部大会
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

抗がん剤耐性克服を志向したKeap1-リン酸化p62タンパク質間相互作用阻害剤の創薬研究

Speaker
○安田大輔、中島真央、髙橋恭子、大江知之、一村義信、小松雅明、今村理世、小島宏建、岡部隆義、長野哲雄、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.05.17 - 2018.05.17
Organizer
第71回日本酸化ストレス学会
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

抗酸化活性を有する非フェノール型尿酸アナログの創製

Speaker
伊藤理人、比留川史也、○髙橋恭子、中村成夫、大江知之、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.03.25 - 2018.03.25
Organizer
日本薬学会第138年会
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

医薬品としての物性向上を目指したKeap1-リン酸化p62結合阻害剤の創製

Speaker
○中島真央、安田大輔、大江知之、高橋恭子、小松雅明、一村義信、今村理世、小島宏建、岡部隆義、長野哲雄、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.03.25 - 2018.03.25
Organizer
日本薬学会第138年会
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

グルクロン酸抱合経由の代謝活性化を回避したジクロフェナク類縁体の創製

Speaker
山田晶子、○大江知之、小川真依、髙橋恭子、中村成夫、増野匡彦
Conference Title
[Conference Category Domestic presentation] Dates 2018.03.25 - 2018.03.25
Organizer
日本薬学会第138年会
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

ADMET研究と融合したアカデミア創薬

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2018.03.10 - 2018.03.10
Invitation Status
With
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (invited, special)

抗 HIV 薬を目指した新規ピリジニウム型フラーレン誘導体の創製

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.10.26 - 2017.10.26
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

HIV 逆転写酵素阻害活性を有するジドブジン結合型新規フラーレン誘導体の創製

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.09.16 - 2017.09.16
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

代謝活性化を回避した新規ベンズブロマロン類縁体の合成およびその毒性評価

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.09.16 - 2017.09.16
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

ADMET研究と創薬化学を融合した新しいアカデミア創薬

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.09.16 - 2017.09.16
Invitation Status
With
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Symposium, workshop panel (nominated)

抗がん薬を⽬指した新規ピリジニウム型C60 誘導体の創製

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.09.12 - 2017.09.12
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Oral presentation (general)

薬学共用試験CBT―2016 年度結果について

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.09.03 - 2017.09.03
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

2016年度薬学共用試験報告

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.08.18 - 2017.08.18
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation

HCVポリメラーゼ/プロテアーゼ二重阻害活性を有するフラーレン誘導体の細胞内HCV複製阻害及び酸化ストレス抑制効果

Speaker
MASHINO Tadahiko
Conference Title
[Conference Category Domestic presentation] Dates 2017.03.27 - 2017.03.27
Invitation Status
Without
Presentation Format
Domestic presentation
Language of Publication
Japanese
Conference Category
Poster presentation